23076-35-9, Xylazine hydrochloride
Ts'ebeliso ea Xylazine hydrochloride
Xylazine HydrochlorideSepheo: Adrenergic ReceptorXylazine ke setlhare se sebelisetsoang sedation, thethebatso, phomolo ea mesifa le analgesia liphoofolong tse kang lipere, likhomo le liphoofolo tse ling tse anyesang tseo e seng batho. Analog ea clonidine, ke agonist sehlopheng sa α2 sa adrenergic receptor. Xylazine e sa tsoa hlaha e le setlhare sa boithabiso, haholoholo Puerto Rico [1]. Tsamaiso ea xylazine (0.17 mg / kg ea boima ba 'mele, e hlapolotsoeng ho ea ho molumo oa 10-ml, e sebelisa 0.9% NaCl) e hlohlellelitse lihora tse ka bang 2.5 tsa analgesia ea lehae ntle le litlamorao tse hlakileng. Mefuta e phahameng ea xylazine e bakile ataxia ea maoto a ka morao a bonolo. Tsamaiso ea lidocaine e bakile nako e tšoanang ea analgesia, e nang le leoto le leholo le ka morao la ataxia (100% incidence). Re fihletse qeto ea hore xylazine e fanoeng ke ente ea epidural e fella ka analgesia e sireletsehileng, e sebetsang ea perineal analgesia lipere [2].
Xylazine hydrochloride Ketsahalo ea Bioloji
Tlhaloso | Xylazine Hydrochloride ke sehlopha sa α2 sa adrenergic receptor agonist. Sepheo: Adrenergic ReceptorXylazine ke setlhare se sebelisetsoang sedation, thethebatso, phomolo ea mesifa le analgesia liphoofolong tse kang lipere, likhomo le liphoofolo tse ling tse anyesang tseo e seng batho. Analog ea clonidine, ke agonist sehlopheng sa α2 sa adrenergic receptor. Xylazine e sa tsoa hlaha e le setlhare sa boithabiso, haholoholo Puerto Rico [1]. Tsamaiso ea xylazine (0.17 mg / kg ea boima ba 'mele, e hlapolotsoeng ho ea ho molumo oa 10-ml, e sebelisa 0.9% NaCl) e hlohlellelitse lihora tse ka bang 2.5 tsa analgesia ea lehae ntle le litlamorao tse hlakileng. Mefuta e phahameng ea xylazine e bakile ataxia ea maoto a ka morao a bonolo. Tsamaiso ea lidocaine e bakile nako e tšoanang ea analgesia, e nang le leoto le leholo le ka morao la ataxia (100% incidence). Re fihletse qeto ea hore xylazine e fanoeng ke ente ea epidural e fella ka analgesia e sireletsehileng, e sebetsang ea perineal analgesia lipere [2]. |
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Catalog e Amanang | |
Litšupiso | [1]. Reyes, JC, et al., Ho hlaha ha xylazine e le sethethefatsi se secha sa tlhekefetso le litlamorao tsa bophelo bo botle har'a basebelisi ba lithethefatsi Puerto Rico. J Bophelo bo Botle ba Litoropo, 2012. 89 (3): leq. 519-26.[2]. Hsu, WH, khatello ea maikutlo e bakoang ke Xylazine le ho hanyetsana ha eona ke alpha adrenergic block agents. J Pharmacol Exp Ther, 1981. 218 (1): leq. 188-92. |
Lik'hemik'hale le Thepa ea 'mele
Ho teteana | 1.15g / cm3 |
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Ntlha ea ho belisoa | 334.2ºC ho 760mmHg |
Qhibiliha Point | 150-164? C (qeto.) |
Foromo ea Limolek'hule | C12H17ClN2S |
Boima ba limolek'hule | EA-256.795 |
Flash Point | 15º.9 ° C |
'Misa o nepahetseng | EA-256.080109 |
PSA | 49.69000 |
LogP | 3.51880 |
Khatello ea Moea | 0.00013mmHg ka 25 ° C |
Boemo ba polokelo | -20 ° C |
Tlhahisoleseling e nang le chefo
TLHALOSO MOTSOALLE
DATA EA KOTSI EA BOPHELOLITLHAKU TSE KOTSI LITLHAHISO
|
Mabitso a tšoanang ka moelelo
BAY 1470 hydrochloride |
Xylazine chloride |
2- (2,6-Dimethylphenylamino) -5,6-dihydro-4H-thiazine hydrochloride |
2 - [(2,6-Dimethylphenyl) amino] -5,6-dihydro-4H-1, 3-thiazine Hydrochloride |
N- (2,6-Dimethylphenyl) -5,6-dihydro-4H-1,3-thiazin-2-amine hydrochloride (1: 1) |
BAY VA 1470 |
EINECS 245-417-0 |
4H-1,3-Thiazin-2-amine, N- (2, 6-dimethylphenyl) -5,6-dihydro-, hydrochloride (1: 1) |
Celactal |
N- (2,6-Dimethylphenyl) -5, 6-dihydro-4H-1,3-thiazin-2-amine hydrochloride |
Xylazine HCl |
MFCD00058196 |


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